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Search Results for " prolyl oligopeptidase "

ターゲット

9

阻害剤

6

天然化合物

1

リコンビナントタンパク質

カタログ番号 製品名 別名 ターゲット
T8657 KYP-2047 Others
KYP-2047 is a very potent, selective Prolyl oligopeptidase (POP) inhibitor.
T9855 BR102910  4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]- Others
BR102910 (4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-) is a selective inhibitor of fibroblast activated protein (FAP).
T61622 PREP inhibitor-1 Others
PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.
T21011 Buspirone Buspirone free base,Ansial 5-HT Receptor
Buspirone (Buspirone free base) is an azaspiro compound which has a role as an anxiolytic drug, a sedative, a serotonergic agonist and an EC 3.4.21.26 (prolyl oligopeptidase) inhibitor.
T7890 SP-13786 UAMC-1110 Others
SP-13786 (UAMC-1110) is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM).
T78619 Z-Pro-Pro-CHO Prolyl Endopeptidase (PREP)
Z-Pro-Pro-CHO acts as a prolyl oligopeptidase inhibitor with half-maximal inhibitory concentrations (IC50) of 0.16 μM for human prolyl oligopeptidase and 0.01 μM for Schistosoma mansoni prolyl oligopeptidase [1].
T61995 Y-29794
Y-29794 (Compound 2) is a potent, covalent inhibitor of prolyl oligopeptidase (POP) (Ki= 0.95 nM). Y-29794 has research value in neurodegenerative diseases and cancer.
T62534 POP-IN-2
POP-IN-2 (Compound 7k) is a potent, covalently bound inhibitor of prolyl oligopeptidase (POP) (Ki: 6 nM).POP-IN-2 can be used in neurodegenerative disease and cancer research.
T69603 BR103354
BR103354 is a novel fibroblast activation protein (FAP) inhibitor with anti-diabetic and anti-steatotic effects. BR103354 inhibited FAP with an IC50 value of 14 nM, showing high selectivity against dipeptidyl peptidase (...
カタログ番号 製品名 別名 ターゲット
TN4442 Linderene acetate Prolyl Endopeptidase (PREP)
Linderene acetate is a competitive inhibitor against Prolyl endopeptidase.
T2717 Salidroside Rhodioloside Apoptosis , mTOR
Salidroside (Rhodioloside) is a bioactive phenolic glycoside compound isolated from Rhodiola crenulata. It is a prolyl endopeptidase Inhibitor.
T3891 Oroxylin A-7-O-glucuronide Oroxylin A Glucoronide,Oroxyloside,Oroxylin A 7-O-beta-D-glucuronide Others
Oroxylin A-7-O-glucuronide (Oroxylin A Glucoronide) and wogonoside should also be served as the chemical markers together with baicalin for the quality control of herbs and proprietary traditional Chinese medicine (PTCM)...
T2S0618 β-Elemonic Acid 3-oxo Tirucallic Acid,Beta-Elemonic acid,3-Oxotirucallenoic Acid,Elemadienonic Acid Apoptosis , Reactive Oxygen Species , COX
β-Elemonic Acid (3-Oxotirucallenoic Acid) exhibits anti-inflammatory effects. Beta-Elemonic acid inhibits proliferation by inducing hypoploid cells and cell apoptosis, the anticancer effects of beta-Elemonic acid are rel...
TN3714 (-)-Corypalmine Corypalmine Antifection
Corypalmine (IC50=128.0±10.5 uM) can inhibit prolyl oligopeptidase. (-)-Corypalmine shows inhibition activity against spore germination of some fungi.
TN4426 Leojaponin AChR
Leojaponin is a prolyl oligopeptidase (POP) inhibitor. Leojaponin exhibits significant cytoprotective activities against glutamate-induced toxicity at concentrations ranging from 0.1 microm to 10 microm.

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPY-03269 Prolyl Endopeptidase Protein, Mouse, Recombinant (His) Mouse Baculovirus Insect Cells
Prolyl endopeptidase, also known as PREP, belongs to a distinct class of serine peptidases. It is a large cytosolic enzyme which was first described in the cytosol of rabbit brain as an oligopeptidase. Prolyl endopeptida...